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Educational purposes only. Not medical advice. Consult healthcare professionals before use.

Healing & Recovery
Preclinical

Epitalon

Epitalon

Also known as: Epithalon, Epithalone, AGAG, Ala-Glu-Asp-Gly

Overview

Key Facts

Primary Goal: Research and therapeutic applications of Epitalon

Stimulates pinealocytes to restore melatonin synthesis and secretion. Reactivates genes involved in circadian clock regulation.

Dosing Information

Half-Life

~2-3 hours

Typical Dose

5–10 mg

Frequency

Once daily for 10-20 day cycles

Cycle Length

10-20 days on, 4-6 months off

Administration Routes:
subcutaneousintramuscular

Benefits

  • Restores age-depleted melatonin production for natural sleep regulation
  • Normalizes circadian rhythm in elderly individuals
  • Activates telomerase to lengthen telomeres (anti-ageing crossover)
  • Improves sleep onset and sleep quality through pineal gland support
  • Supports immune function and neuroendocrine balance

Side Effects

Mild injection site irritationmild
Drowsiness (related to melatonin upregulation)mild
Headache (uncommon)mild

Mechanism of Action

1

Stimulates pinealocytes to restore melatonin synthesis and secretion

2

Reactivates genes involved in circadian clock regulation

3

Activates telomerase enzyme (hTERT) for anti-ageing effects

4

Enhances antioxidant defence enzymes (SOD, catalase) to reduce oxidative sleep disruption

Contraindications

Do not use this peptide if any of the following apply:

  • Active cancer (telomerase activation could theoretically promote tumour growth)
  • Autoimmune conditions without medical supervision
  • Pregnancy or breastfeeding

Storage & Reconstitution

Unreconstituted (Powder)

Temperature2–8°C (36–46°F) or -20°C (-4°F) for long-term
DurationUp to 3 months

Reconstituted (Mixed)

Temperature2–8°C (36–46°F)
Duration2-4 weeks

Research Summary

Preclinical

Developed by Professor Vladimir Khavinson at the St. Petersburg Institute of Bioregulation and Gerontology. A key study in elderly patients (ages 60-80) demonstrated that Epitalon restored evening melatonin peaks to levels resembling those of younger adults, with corresponding improvements in sleep quality and daytime alertness. The 15-year longitudinal study showed improved immune function, cardiovascular health, and endocrine balance alongside the sleep benefits. Its dual role in melatonin restoration and telomere elongation makes it uniquely positioned among sleep-supportive peptides.

Frequently Asked Questions

Common questions about Epitalon

UK-Specific Information

Exclusive data points and guidance for UK residents using Epitalon

UK Lab Testing

UK Lab Testing

Recommended labs: Medichecks, Thriva (£89-£149 for peptide safety panel)

Why this matters: UK-specific lab testing guidance not available on US competitor sites

Commonly Stacked With

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